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服务
产品  
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SHU 9119
| 名称
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SHU 9119
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| 别名
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| 序列（单字母缩写）
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| 序列（三字母缩写）
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Ac-Nle-cyclo[Asp-His-D-Nal(2')-Arg-Trp-Lys]-NH2
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| C-端
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Amidation
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| 化学桥
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Asp2-Lys7
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| 基本描述
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The efficacy and specificity of SHU-9119 as an MC3/MC4 receptor antagonist in the rat was first validated in vitro and in vivo. In vitro, in heterologous cells expressing either rat MC3-R or MC4-R, the major MCR subtypes expressed in brain, SHU-9119 showed no intrinsic agonism.
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| 溶解度
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Soluble in water. The contents of this vial have been accurately determined. Both the stopper and the vial have been siliconized. Do not attempt to weight out a smaller portion of the contents.
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| 分子量
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1074.230
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| 化学式
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C54H71N15O9
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| 纯度
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> 95%
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| 存储条件
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Storage at -20°C. Keep tightly closed.
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| N-端
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Acetylation
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| 注释
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Antagonist of rat MC3 and mouse MC4 receptors.
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